Mo Haskali

A New Turn in Peptide-Based Imaging Agents: Foldamers Afford Improved Theranostics Targeting Cholecystokinin-2 Receptor-Positive Cancer.

Alicia Corlett, Marc-Antoine Sani, Jessica Van Zuylekom, Ching-Seng Ang, Elisabeth von Guggenberg, Carleen Cullinane, Benjamin Blyth, Rodney J Hicks, Peter D Roselt, Philip E Thompson, Craig A Hutton, Mohammad B Haskali

Journal article  |  2021  |  Journal of Medicinal Chemistry

Proteins adopt unique folded secondary and tertiary structures that are responsible for their remarkable biological properties. Th..

Bivalent Inhibitors of Prostate-Specific Membrane Antigen Conjugated to Desferrioxamine B Squaramide Labeled with Zirconium-89 or Gallium-68 for Diagnostic Imaging of Prostate Cancer

Asif Noor, Jessica K Van Zuylekom, Stacey E Rudd, Kelly Waldeck, Peter D Roselt, Mohammad B Haskali, Michael P Wheatcroft, Eddie Yan, Rodney J Hicks, Carleen Cullinane, Paul S Donnelly

Journal article  |  2020  |  Journal of Medicinal Chemistry

Prostate-specific membrane antigen (PSMA) is a carboxypeptidase that is overexpressed in prostate cancer and is an excellent candi..

Gallium Fluoride Complexes with Acyclic Bispicolinic Ligands as Potential New Fluorine-18 Labelled Imaging Agents

HuiJing Koay, Mohammad B Haskali, Peter D Roselt, Jonathan M White, Paul S Donnelly

Journal article  |  2020  |  European Journal of Inorganic Chemistry

4-Nitrophenyl activated esters are superior synthons for indirect radiofluorination of biomolecules

Mohammad B Haskali, Ashleigh L Farnsworth, Peter D Roselt, Craig A Hutton

Journal article  |  2020  |  MedChemComm

PET ligands [F-18]LSN3316612 and [C-11]LSN3316612 quantify O-linked-beta-N-acetyl-glucosamine hydrolase in the brain

Shuiyu Lu, Mohammad B Haskali, Kevin M Ruley, Nicolas J-F Dreyfus, Susan L DuBois, Soumen Paul, Jeih-San Liow, Cheryl L Morse, Aneta Kowalski, Robert L Gladding, Jeremy Gilmore, Adrian J Mogg, S Michelle Morin, Peter J Lindsay-Scott, J Craig Ruble, Nancy A Kant, Sergey Shcherbinin, Vanessa N Barth, Michael P Johnson, Maria Cuadrado, et al.

Journal article  |  2020  |  Science Translational Medicine

A Cu-64/Cu-67 bifunctional PSMA ligand as a theranostic for prostate cancer

Lachlan McInnes, Nicholas Zia, Carleen Cullinane, Jessica Van Zuylekom, Susan Jackson, Jon Stoner, Mohammad Haskali, Peter Roselt, Ellen Van Dam, Matthew Harris, Rodney Hicks, Paul Donnelly

Conference Proceedings  |  2020  |  JOURNAL OF NUCLEAR MEDICINE

PET quantification of brain O-GlcNAcase with [F-18]LSN3316612 in healthy human volunteers

Jae-Hoon Lee, Jeih-San Liow, Soumen Paul, Cheryl L Morse, Mohammad B Haskali, Lester Manly, Sergey Shcherbinin, J Craig Ruble, Nancy Kant, Emily C Collins, Hugh N Nuthall, Paolo Zanotti-Fregonara, Sami S Zoghbi, Victor W Pike, Robert B Innis

Journal article  |  2020  |  EJNMMI Research

Radiosynthesis and preliminary in vivo evaluation of F-18-labelled glycosylated duramycin peptides for imaging of phosphatidylethanolamine during apoptosis

Mohammad B Haskali, Delphine Denoyer, Peter D Roselt, Rodney J Hicks, Craig A Hutton

Journal article  |  2019  |  RSC Medicinal Chemistry

[18F]-Labelled duramycin derivatives incorporating hydrophilic aminogalacturonic acid moieties were prepared as tracers for in viv..

A Bivalent Inhibitor of Prostate Specific Membrane Antigen Radiolabeled with Copper-64 with High Tumor Uptake and Retention

Nicholas A Zia, Carleen Cullinane, Jessica K Van Zuylekom, Kelly Waldeck, Lachlan E McInnes, Gojko Buncic, Mohammad B Haskali, Peter D Roselt, Rodney J Hicks, Paul S Donnelly

Journal article  |  2019  |  Angewandte Chemie International Edition

Automated preparation of clinical grade [68Ga]Ga-DOTA-CP04, a cholecystokinin-2 receptor agonist, using iPHASE MultiSyn synthesis platform.

Mohammad B Haskali, Peter D Roselt, David Binns, Amit Hetsron, Stan Poniger, Craig A Hutton, Rodney J Hicks

Journal article  |  2019  |  EJNMMI Radiopharmacy and Chemistry

BACKGROUND: Gallium-68 ([68Ga]Ga) labelled radiopharmaceuticals have become a valuable tool in clinical practice using Positron Em..