Daniel Priebbenow

Discovery of Acylsulfonohydrazide-Derived Inhibitors of the Lysine Acetyltransferase, KAT6A, as Potent Senescence-Inducing Anti-Cancer Agents

Daniel L Priebbenow, David J Leaver, Nguyen Nghi, Benjamin Cleary, H Rachel Lagiakos, Julie Sanchez, Lian Xue, Fei Huang, Yuxin Sun, Prashant Mujumdar, Ramesh Mudududdla, Swapna Varghese, Silvia Teguh, Susan A Charman, Karen L White, David M Shackleford, Kasiram Katneni, Matthew Cuellar, Jessica M Strasser, Jayme L Dahlin, et al.

Journal article  |  2020  |  Journal of Medicinal Chemistry

A high-throughput screen designed to discover new inhibitors of histone acetyltransferase KAT6A uncovered CTX-0124143 (1), a uniqu..

Silicon-Derived Singlet Nucleophilic Carbene Reagents in Organic Synthesis

Daniel L Priebbenow

Journal article  |  2020  |  Advanced Synthesis & Catalysis

Insights into the Stability of Siloxy Carbene Intermediates and Their Corresponding Oxocarbenium Ions

Daniel L Priebbenow

Journal article  |  2019  |  The Journal of Organic Chemistry

Discovery of Benzoylsulfonohydrazides as Potent Inhibitors of the Histone Acetyltransferase KAT6A

David J Leaver, Benjamin Cleary, Nguyen Nghi, Daniel L Priebbenow, H Rachel Lagiakos, Julie Sanchez, Lian Xue, Fei Huang, Yuxin Sun, Prashant Mujumdar, Ramesh Mudududdla, Swapna Varghese, Silvia Teguh, Susan A Charman, Karen L White, Kasiram Katneni, Matthew Cuellar, Jessica M Strasser, Jayme L Dahlin, Michael A Walters, et al.

Journal article  |  2019  |  Journal of Medicinal Chemistry

A high-throughput screen for inhibitors of the histone acetyltransferase, KAT6A, led to identification of an aryl sulfonohydrazide..

Substituted Pyridazin-3(2H)-ones as Highly Potent and Biased Formyl Peptide Receptor Agonists

Girdhar Singh Deora, Cheng Xue Qin, Elizabeth A Vecchio, Aaron J Debono, Daniel L Priebbenow, Ryan M Brady, Julia Beveridge, Silvia C Teguh, Deo Minh, Lauren T May, Guy Krippner, Rebecca H Ritchie, Jonathan B Baell

Journal article  |  2019  |  Journal of Medicinal Chemistry

New synthetic approaches towards analogues of bedaquiline

Daniel L Priebbenow, Lisa Barbaro, Jonathan B Baell

Journal article  |  2016  |  Organic & Biomolecular Chemistry

Iron-Catalyzed Acylative Dealkylation of N-Alkylsulfoximines

Philip Lamers, Daniel L Priebbenow, Carsten Bolm

Journal article  |  2015  |  European Journal of Organic Chemistry

Regio- and Stereoselective Iodoacyloxylations of Alkynes

Daniel L Priebbenow, Robert W Gable, Jonathan Baell

Journal article  |  2015  |  The Journal of Organic Chemistry

The Synthesis of Chiral Benzothiazine and Thiazinoquinoline Derivatives

Long Wang, Daniel L Priebbenow, Xiao Yun Chen, Fang-Fang Pan, Carsten Bolm

Journal article  |  2015  |  European Journal of Organic Chemistry

N-Arylations of Sulfoximines with 2-Arylpyridines by Copper-Mediated Dual N-H/C-H Activation

Long Wang, Daniel L Priebbenow, Wanrong Dong, Carsten Bolm

Journal article  |  2014  |  Organic Letters

C-H Activation of Methyl Arenes in the MnO2-Mediated Aroylation of N-Chlorosulfoximines

Daniel L Priebbenow, Carsten Bolm

Journal article  |  2014  |  Organic Letters

Photochemical Intermolecular Silylacylations of Electron-Deficient Internal Alkynes

Peter Becker, Daniel L Priebbenow, Hui-Jun Zhang, Ramona Pirwerdjan, Carsten Bolm

Journal article  |  2014  |  The Journal of Organic Chemistry

Acylsilanes in Rhodium(III)-Catalyzed Directed Aromatic C-H Alkenylations and Siloxycarbene Reactions with C-C Double Bonds

Peter Becker, Daniel L Priebbenow, Ramona Pirwerdjan, Carsten Bolm

Journal article  |  2014  |  Angewandte Chemie International Edition

Copper-Catalyzed Oxidative Decarboxylative Couplings of Sulfoximines and Aryl Propiolic Acids

Daniel L Priebbenow, Peter Becker, Carsten Bolm

Journal article  |  2013  |  Organic Letters

Exploring the Reactivity of N-Alkynylated Sulfoximines: [2 2]-Cycloadditions

Ramona Pirwerdjan, Daniel L Priebbenow, Peter Becker, Philip Lamers, Carsten Bolm

Journal article  |  2013  |  Organic Letters

Copper-Catalyzed Synthesis of alpha-Thioaryl Carbonyl Compounds Through S-S and C-C Bond Cleavage

Liang-Hua Zou, Daniel L Priebbenow, Long Wang, Jakob Mottweiler, Carsten Bolm

Journal article  |  2013  |  Advanced Synthesis & Catalysis

The Disubstitution of Acetals to Prepare ,-Bis(aryl) -Keto Esters

Daniel L Priebbenow, Liang-Hua Zou, Peter Becker, Carsten Bolm

Journal article  |  2013  |  European Journal of Organic Chemistry

The Copper-Catalyzed Oxidative N-Acylation of Sulfoximines

Long Wang, Daniel L Priebbenow, Liang-Hua Zou, Carsten Bolm

Journal article  |  2013  |  Advanced Synthesis & Catalysis

Mild Copper-Mediated Direct Oxidative Cross-Coupling of 1,3,4-Oxadiazoles with Polyfluoroarenes by Using Dioxygen as Oxidant

Liang-Hua Zou, Jakob Mottweiler, Daniel L Priebbenow, Jun Wang, Jan Alexander Stubenrauch, Carsten Bolm

Journal article  |  2013  |  Chemistry - A European Journal

CH(3)CN and O(2) do the trick! A copper-mediated direct oxidative cross-coupling of 2-(het)aryl-1,3,4-oxadiazoles with polyhaloare..

The rhodium-catalysed synthesis of pyrrolidinone-substituted (trialkylsilyloxy)acrylic esters

Daniel L Priebbenow, Carsten Bolm

Journal article  |  2013  |  RSC Advances

Copper-Catalyzed Oxidative Cross-Coupling of Sulfoximines and Alkynes

Long Wang, He Huang, Daniel L Priebbenow, Fang-Fang Pan, Carsten Bolm

Journal article  |  2013  |  Angewandte Chemie International Edition

Acylsilanes: valuable organosilicon reagents in organic synthesis

Hui-Jun Zhang, Daniel L Priebbenow, Carsten Bolm

Journal article  |  2013  |  Chemical Society Reviews

Recent advances in the Willgerodt-Kindler reaction

Daniel L Priebbenow, Carsten Bolm

Journal article  |  2013  |  Chemical Society Reviews

Asymmetric induction in domino Heck-aza-Michael reactions

Daniel L Priebbenow, Scott G Stewart, Frederick M Pfeffer

Journal article  |  2012  |  Tetrahedron Letters

A One-Pot, Three-Component Approach to Functionalised Tetrahydroisoquinolines Using Domino Heck-aza-Michael Reactions

Daniel L Priebbenow, Frederick M Pfeffer, Scott G Stewart

Journal article  |  2011  |  European Journal of Organic Chemistry

A general approach to N-heterocyclic scaffolds using domino Heck-aza-Michael reactions

Daniel L Priebbenow, Scott G Stewart, Frederick M Pfeffer

Journal article  |  2011  |  Organic & Biomolecular Chemistry

Domino Heck-Aza-Michael Reactions: Efficient Access to 1-Substituted Tetrahydro-beta-carbolines

Daniel L Priebbenow, Luke C Henderson, Frederick M Pfeffer, Scott G Stewart

Journal article  |  2010  |  The Journal of Organic Chemistry

Investigations into the Stability of Siloxy Carbene Intermediates and the Corresponding Oxocarbenium Ions

Daniel Priebbenow

Journal article

This report describes an investigation using dispersion-corrected DFT into the structures and stabilities of siloxy carbenes. Silo..