Daniel Priebbenow

Discovery of Acylsulfonohydrazide-Derived Inhibitors of the Lysine Acetyltransferase, KAT6A, as Potent Senescence-Inducing Anti-Cancer Agents

Daniel L Priebbenow, David J Leaver, Nguyen Nghi, Benjamin Cleary, H Rachel Lagiakos, Julie Sanchez, Lian Xue, Fei Huang, Yuxin Sun, Prashant Mujumdar, Ramesh Mudududdla, Swapna Varghese, Silvia Teguh, Susan A Charman, Karen L White, David M Shackleford, Kasiram Katneni, Matthew Cuellar, Jessica M Strasser, Jayme L Dahlin, et al.

Journal article  |  2020  |  Journal of Medicinal Chemistry

A high-throughput screen designed to discover new inhibitors of histone acetyltransferase KAT6A uncovered CTX-0124143 (1), a uniqu..

Silicon-Derived Singlet Nucleophilic Carbene Reagents in Organic Synthesis

Daniel L Priebbenow

Journal article  |  2020  |  Advanced Synthesis & Catalysis

Insights into the Stability of Siloxy Carbene Intermediates and Their Corresponding Oxocarbenium Ions

Daniel L Priebbenow

Journal article  |  2019  |  The Journal of Organic Chemistry

Discovery of Benzoylsulfonohydrazides as Potent Inhibitors of the Histone Acetyltransferase KAT6A

David J Leaver, Benjamin Cleary, Nguyen Nghi, Daniel L Priebbenow, H Rachel Lagiakos, Julie Sanchez, Lian Xue, Fei Huang, Yuxin Sun, Prashant Mujumdar, Ramesh Mudududdla, Swapna Varghese, Silvia Teguh, Susan A Charman, Karen L White, Kasiram Katneni, Matthew Cuellar, Jessica M Strasser, Jayme L Dahlin, Michael A Walters, et al.

Journal article  |  2019  |  Journal of Medicinal Chemistry

A high-throughput screen for inhibitors of the histone acetyltransferase, KAT6A, led to identification of an aryl sulfonohydrazide..

Substituted Pyridazin-3(2H)-ones as Highly Potent and Biased Formyl Peptide Receptor Agonists

Girdhar Singh Deora, Cheng Xue Qin, Elizabeth A Vecchio, Aaron J Debono, Daniel L Priebbenow, Ryan M Brady, Julia Beveridge, Silvia C Teguh, Deo Minh, Lauren T May, Guy Krippner, Rebecca H Ritchie, Jonathan B Baell

Journal article  |  2019  |  Journal of Medicinal Chemistry

New synthetic approaches towards analogues of bedaquiline

Daniel L Priebbenow, Lisa Barbaro, Jonathan B Baell

Journal article  |  2016  |  Organic & Biomolecular Chemistry

Iron-Catalyzed Acylative Dealkylation of N-Alkylsulfoximines

Philip Lamers, Daniel L Priebbenow, Carsten Bolm

Journal article  |  2015  |  European Journal of Organic Chemistry

Regio- and Stereoselective Iodoacyloxylations of Alkynes

Daniel L Priebbenow, Robert W Gable, Jonathan Baell

Journal article  |  2015  |  The Journal of Organic Chemistry

The Synthesis of Chiral Benzothiazine and Thiazinoquinoline Derivatives

Long Wang, Daniel L Priebbenow, Xiao Yun Chen, Fang-Fang Pan, Carsten Bolm

Journal article  |  2015  |  European Journal of Organic Chemistry

N-Arylations of Sulfoximines with 2-Arylpyridines by Copper-Mediated Dual N-H/C-H Activation

Long Wang, Daniel L Priebbenow, Wanrong Dong, Carsten Bolm

Journal article  |  2014  |  Organic Letters