Dr. Helene Jousset Sabroux
Honorary
Medical Biology (W.E.H.I.)
10 Scholarly works
0 Projects
HIGHLIGHTS
2020
Journal article
Discovery of Acylsulfonohydrazide-Derived Inhibitors of the Lysine Acetyltransferase, KAT6A, as Potent Senescence-Inducing Anti-Cancer Agents
DOI: 10.1021/acs.jmedchem.9b020712019
Journal article
Viral MLKL Homologs Subvert Necroptotic Cell Death by Sequestering Cellular RIPK3
DOI: 10.1016/j.celrep.2019.08.0552019
Journal article
Discovery of Benzoylsulfonohydrazides as Potent Inhibitors of the Histone Acetyltransferase KAT6A
DOI: 10.1021/acs.jmedchem.9b006652019
Journal article
Identification of 5-Substituted 2-Acylaminothiazoles That Activate Tat-Mediated Transcription in HIV-1 Latency Models
DOI: 10.1021/acs.jmedchem.9b004622019
Journal article
Therapeutic Effects of a TANK-Binding Kinase 1 Inhibitor in Germinal Center-Driven Collagen-Induced Arthritis
DOI: 10.1002/art.406702018
Journal article
Enhanced antimalarial activity of plasmepsin V inhibitors by modification of the P-2 position of PEXEL peptidomimetics
DOI: 10.1016/j.ejmech.2018.05.0222017
Journal article
Design, Synthesis, and Biological Activity of 1,2,3-Triazolobenzodiazepine BET Bromodomain Inhibitors
DOI: 10.1021/acsmedchemlett.7b00389
RECENT SCHOLARLY WORKS
2017
Journal article
Colorectal Cancer Cell Line Proteomes Are Representative of Primary Tumors and Predict Drug Sensitivity
DOI: 10.1053/j.gastro.2017.06.0082017
Journal article
Optimization of 2-Anilino 4-Amino Substituted Quinazolines into Potent Antimalarial Agents with Oral in Vivo Activity
DOI: 10.1021/acs.jmedchem.6b016732016
Journal article
Exploration of the P-3 region of PEXEL peptidomimetics leads to a potent inhibitor of the Plasmodium protease, plasmepsin V
DOI: 10.1016/j.bmc.2016.03.027