Journal article

A randomized, double-blind, placebo-controlled phase 1b/2 study of ralimetinib, a p38 MAPK inhibitor, plus gemcitabine and carboplatin versus gemcitabine and carboplatin for women with recurrent platinum-sensitive ovarian cancer

I Vergote, F Heitz, P Buderath, M Powell, J Sehouli, CM Lee, A Hamilton, J Fiorica, KN Moore, M Teneriello, L Golden, W Zhang, C Pitou, R Bell, R Campbell, DL Farrington, K Bell-McGuinn, RM Wenham

Gynecologic Oncology | ACADEMIC PRESS INC ELSEVIER SCIENCE | Published : 2020

Abstract

Objective: This phase 1b/2 clinical trial (NCT01663857) evaluated the efficacy of ralimetinib in combination with gemcitabine (G) and carboplatin (C), followed by maintenance ralimetinib, for patients with recurrent platinum-sensitive epithelial ovarian cancer. Methods: Phase 1b was to determine the recommended phase 2 dose (RP2D) of ralimetinib administered Q12H on Days 1–10 (q21d) in combination with G (1000 mg/m2, Days 3 and 10) and C (AUC 4, Day 3) for six cycles. In phase 2, patients were randomized double-blind 1:1 to ralimetinib (R)+GC or placebo (P)+GC, for six cycles, followed by ralimetinib 300 mg Q12H or placebo on Days 1–14, q28d. Results: 118 patients received at least one dose ..

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University of Melbourne Researchers