Journal article

Pharmacokinetics of chloroquine and monodesethylchloroquine in pregnancy

HA Karunajeewa, S Salman, I Mueller, F Baiwog, S Gomorrai, I Law, M Page-Sharp, S Rogerson, P Siba, KF Ilett, TME Davis

Antimicrobial Agents and Chemotherapy | AMER SOC MICROBIOLOGY | Published : 2010

Abstract

In order to determine the pharmacokinetic disposition of chloroquine (CQ) and its active metabolite, desethylchloroquine (DECQ), when administered as intermittent presumptive treatment in pregnancy (IPTp) for malaria, 30 Papua New Guinean women in the second or third trimester of pregnancy and 30 age-matched nonpregnant women were administered three daily doses of 450 mg CQ (8.5 mg/kg of body weight/day) in addition to a single dose of sulfadoxine-pyrimethamine. For all women, blood was taken at baseline; at 1, 2, 4, 6, 12, 18, 24, 30, 48, and 72 h posttreatment; and at 7, 10, 14, 28, and 42 days posttreatment. Plasma was subsequently assayed for CQ and DECQ by high-performance liquid chroma..

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University of Melbourne Researchers

Grants

Awarded by National Health and Medical Research Council of Australia


Funding Acknowledgements

The study was funded by the National Health and Medical Research Council of Australia (grant 458555). T. M. E. D. is supported by a National Health and Medical Research Council of Australia Practitioner Fellowship.